Modulation of Kv3.4 channel N-type inactivation by protein kinase C shapes the action potential in dorsal root ganglion neurons.

Authors:
Ritter DM, Ho C, O'Leary ME, Covarrubias M.
In:
Source: J Physiol
Publication Date: (2012)
Issue: 590(Pt 1): 145-61
Research Area:
Neurobiology
Cells used in publication:
Dorsal root gang. (DRG), rat
Species: rat
Tissue Origin: brain
Platform:
4D-Nucleofector® X-Unit
Experiment

Approximately 2×106 dissociated rat DRG neurons were transfected with 40 pmol of rat Kv3.4 (KCNC4) siRNA or control siRNA-A (Santa Cruz Biotechnology, Santa Cruz, CA,USA) using theAmaxaNucleofector-II system(Lonza; programme G-013 and Rat Neuron Nucleofector Kit) or 4D-Nucleofector system (Lonza; programme DC-100 and P3 Primary Cell Kit). Immediately after transfection, neurons were allowed to recover for 10 min at 37?C before plating on cover slips. In addition, single-cell qPCR 24 h post-transfection detected Kv3.4 mRNA in 93% of control siRNA-transfected neurons and 60% of Kv3.4 siRNA-transfected neurons.

Abstract

Fast inactivation of heterologously expressed Kv3.4 channels is dramatically slowed upon phosphorylation of the channel's N-terminal (N-type) inactivation gate by protein kinase C (PKC). However, the presence and physiological importance of this exquisite modulation in excitable tissues were unknown. Here, we employed minimally invasive cell-attached patch-clamping, single-cell qPCR and specific siRNAs to unambiguously demonstrate that fast-inactivating Kv3.4 channels underlie a robust high voltage-activated A-type K(+) current (I(AHV)) in nociceptive dorsal root ganglion neurons from 7-day-old rats. We also show that PKC activation with phorbol 12,13-dibutyrate (PDBu) causes a 4-fold slowing of Kv3.4 channel inactivation and, consequently, accelerates the repolarization of the action potential (AP) by 22%, which shortens the AP duration by 14%. G-protein coupled receptor (GPCR) agonists eliminate I(AHV) fast inactivation in a membrane-delimited manner, suggesting a Kv3.4 channel signalling complex. Preincubation of the neurons with the PKC inhibitor bisindolylmaleimide II inhibits the effect of GPCR agonists and PDBu. Furthermore, activation of PKC via GPCR agonists recapitulates the effects of PDBu on the AP. Finally, transfection of the neurons with Kv3.4 siRNA prolongs the AP by 25% and abolishes the GPCR agonist-induced acceleration of the AP repolarization. These results show that Kv3.4 channels help shape the repolarization of the nociceptor AP, and that modulation of Kv3.4 channel N-type inactivation by PKC regulates AP repolarization and duration. We propose that the dramatic modulation of I(AHV) fast inactivation by PKC represents a novel mechanism of neural plasticity with potentially significant implications in the transition from acute to chronic pain.